CAS 1229194-11-9|Edoxaban (tosylate Monohydrate)
Cov mis mos molecular: C31H38ClN7O7S2
Molecular Luj: 720.26
EINECS: 1592732-453-0
Purity: 97% Min.
Pob: 1 g / 5 g / 25 g / 100 g / 1 kg
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Khoom Taw qhia
Taw qhia
Edoxaban yog ib qho kev xaiv ntawm Xa inhibitor qhov ncauj ntsiav tshuaj rau kev tiv thaiv thiab kho cov hlab ntsha sib sib zog nqus thrombosis thiab pulmonary embolism, siv los txo cov kev pheej hmoo ntawm mob stroke thiab cov kab mob embolism hauv cov neeg mob uas tsis yog-valvular atrial fibrillation (NVAF).
Kev ua lom lom
Edoxaban (DU-176b) yog ib qho kev xaiv inhibitor ntawm yam Xa thiab qhov ncauj tshuaj tiv thaiv kab mob.
Kev tshawb fawb hauv vitro
Hauv tib neeg cov ntshav plasma, Edoxaban ntawm {{0}}}.256 thiab 0.508 μM muab ob npaug rau lub sijhawm prothrombin thiab ua kom lub sijhawm thromboplastin ib nrab, feem.
Hauv vivo kev tshawb fawb
Kev tswj hwm qhov ncauj ntawm Edoxaban ua rau muaj zog tiv thaiv-Xa kev ua haujlwm thiab cov tshuaj plasma siab hauv cov nas thiab liab. Hauv vivo, Edoxaban koob tshuaj-nyob ntawm qhov inhibited thrombus tsim nyob rau hauv nas thiab luav qauv ntawm thrombosis.
Cim npe nrov: cas 1229194-11-9,1229194-11-9,edoxaban (tosylate monohydrate), nqe, hais, luv nqi, hauv Tshuag, muag








